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MeCP2 gene therapy ameliorates disease phenotype in mouse model for Pitt Hopkins syndrome
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The cannabinoid CB receptor positive allosteric modulator EC21a exhibits complicated pharmacology
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Synthesis and characterization of chiral 6-azaspiro[2.5]octanes as potent and selective antagonists of the M muscarinic acetylcholine receptor
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Discovery and optimization of a novel CNS penetrant series of mGlu PAMs based on a 1,4-thiazepane core with in vivo efficacy in a preclinical Parkinsonian model
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2020
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Synthesis and SAR of a series of mGlu NAMs based on an ethyl-8-methoxy-4-(4-phenylpiperazin-1-yl)quinoline carboxylate core
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2020
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